SCHEMBL5478290

SCHEMBL5478290

CCCc1c(C(N)=O)cccc1-c1ccccc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
BCAT2 O15382 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADRA2A P08913 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
JAK2 O60674 1/20 0.38
GRM2 Q14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5524497 0.88 PARP1 (0.47) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL21439307 0.86 MAPK8 (0.44) PARP1KEAP1NFE2L2MAPTMEN1
SCHEMBL370726 0.84 MYC (0.45) PARP1BCAT2KEAP1NFE2L2MAPT
SCHEMBL5476512 0.82 BCAT2 (0.59) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL5478916 0.81 MEN1 (0.44) PARP1BCAT2KEAP1NFE2L2MEN1
SCHEMBL2964481 0.81 PARP1 (0.45) PARP1BCAT2KEAP1NFE2L2MAPT
SCHEMBL28784267 0.80 PARP1 (0.50) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL2113823 0.77 NPC1 (0.59) PARP1NPC1RAB9ABCAT2KEAP1
SCHEMBL28204604 0.77 CD38 (0.45) PARP1MAPTMEN1NR1I2LMNA
SCHEMBL5482646 0.77 PPARG (0.45) PARP1NPC1RAB9ABCAT2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763509-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2007-03-21 EP disclosed
WO-2006002474-A1 ALPHA-HELICAL MIMETICS THE WALTER AND ELIZA HALL INSTITUTE OF MEDICAL RESEARCH (AU) 2006-01-12 WO disclosed