SCHEMBL28784875

SCHEMBL28784875

COc1cccc(N2CCN(CCC(=O)NN)CC2)c1

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.69
TP53 P04637 1/20 0.69
THRB P10828 1/20 0.63
DRD2 P14416 2/20 0.62
KCNH2 Q12809 2/20 0.62
DRD4 P21917 4/20 0.62
CACNA1G O43497 2/20 0.61
GFER P55789 3/20 0.60
SMN1; SMN2 Q16637 1/20 0.59
HTR1A P08908 2/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
HTR7 P34969 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2114590 0.85 KCNH2 (0.68) MAPTTP53THRBDRD2KCNH2
SCHEMBL10764516 0.84 HTR1A (0.68) MAPTTHRBDRD2KCNH2CACNA1G
SCHEMBL3198591 0.82 KCNH2 (0.73) MAPTTP53DRD2KCNH2DRD4
Hydrochloric Acid SCHEMBL3212431 0.81 KCNH2 (0.71) MAPTTP53DRD2KCNH2DRD4
SCHEMBL27895258 0.81 KCNH2 (0.76) DRD2KCNH2DRD4CACNA1GHTR1A
SCHEMBL11628265 0.81 DRD2 (0.66) MAPTTP53THRBDRD2KCNH2
SCHEMBL6824119 0.79 KCNH2 (0.76) MAPTDRD2KCNH2GFERSMN1; SMN2
SCHEMBL15743241 0.79 KCNH2 (0.76) MAPTTP53DRD2KCNH2DRD4
SCHEMBL1307825 0.79 KCNH2 (0.76) MAPTDRD2KCNH2GFERSMN1; SMN2
SCHEMBL3045487 0.79 KMT2A (0.56) MAPTDRD2DRD4HTR1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101827828-B 1, 2, 4 -triazole derivatives as serotonergic modulators PROSARIX LTD 2013-02-27 CN disclosed
CN-101827828-A 1, 2, 4 -triazole derivatives as serotonergic modulators PROSARIX LTD 2010-09-08 CN disclosed