SCHEMBL28789909

SCHEMBL28789909

CCOC(=O)c1cccn1-c1cnc(C)c(C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.43
ALDH1A1 P00352 4/20 0.43
SMN1; SMN2 Q16637 6/20 0.42
LMNA P02545 3/20 0.41
RAB9A P51151 5/20 0.40
MAPT P10636 2/20 0.39
KDM4E B2RXH2 4/20 0.38
MAPK1 P28482 1/20 0.38
PDE4D Q08499 1/20 0.38
POLB P06746 1/20 0.38
GABRA1 P14867 3/20 0.38
GABRB2 P47870 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
GABRA2 P47869 2/20 0.38
GLA P06280 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787448 0.78 MAPT (0.54) NPC1ALDH1A1SMN1; SMN2LMNARAB9A
SCHEMBL28960383 0.76 LMNA (0.39) NPC1ALDH1A1SMN1; SMN2LMNARAB9A
SCHEMBL28789880 0.75 SMN1; SMN2 (0.38) NPC1ALDH1A1SMN1; SMN2LMNARAB9A
SCHEMBL31454215 0.72 ALDH1A1 (0.56) NPC1ALDH1A1LMNARAB9AMAPT
SCHEMBL4321608 0.70 MAPT (0.58) NPC1ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL26412819 0.70 CYP2C9 (0.56) NPC1SMN1; SMN2LMNARAB9ACYP1A2
SCHEMBL31454206 0.69 JMJD6 (0.46) NPC1ALDH1A1SMN1; SMN2LMNARAB9A
SCHEMBL2399420 0.68 NPC1 (0.57) NPC1ALDH1A1SMN1; SMN2RAB9AMAPT
SCHEMBL16235806 0.68 SMN1; SMN2 (0.59) ALDH1A1SMN1; SMN2LMNAMAPTKDM4E
SCHEMBL15908738 0.67 TSHR (0.46) ALDH1A1SMN1; SMN2LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114746408-A Alkynyl- (heteroaryl) -carboxamide HCN1 inhibitors 豪夫迈·罗氏有限公司 2022-07-12 CN disclosed