SCHEMBL28791102

SCHEMBL28791102

CC(C)CC(C(=O)O)c1cc(-c2ccccc2)cc(C2CCCN(Cc3ccccc3)C2)c1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CNR2 P34972 1/20 0.41
CYP2D6 P10635 2/20 0.39
DRD2 P14416 3/20 0.39
DRD4 P21917 2/20 0.39
KDM4E B2RXH2 2/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
ALDH1A1 P00352 3/20 0.39
S1PR1 P21453 1/20 0.39
S1PR3 Q99500 1/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2915152 0.95 PSEN1 (0.45) ATML3MBTL1CNR2CYP2D6DRD2
SCHEMBL2903465 0.92 CHRM4 (0.42) ATML3MBTL1CNR2DRD2DRD4
SCHEMBL27894669 0.92 POLB (0.44) ATML3MBTL1CNR2S1PR1S1PR3
SCHEMBL27848935 0.91 PSEN1 (0.40) ATML3MBTL1CYP2D6DRD2DRD4
SCHEMBL27848836 0.91 L3MBTL1 (0.48) ATML3MBTL1CNR2KDM4EALDH1A1
SCHEMBL2903682 0.90 PDE2A (0.41) ATML3MBTL1CNR2DRD2DRD4
SCHEMBL2903669 0.90 PSEN1 (0.39) DRD2DRD4KDM4EPSEN1PSEN2
SCHEMBL2901715 0.88 LMNA (0.41) CNR2KDM4ES1PR1MEN1NPC1
SCHEMBL27848822 0.88 PSEN1 (0.40) KDM4EPSEN1PSEN2APH1BNCSTN
SCHEMBL2922993 0.85 PSEN1 (0.47) L3MBTL1DRD2DRD4PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101903347-B Piperidinyl and piperazinyl modulators of gamma-secretase JANSSEN PHARMACEUTICA NV 2013-03-27 CN disclosed
CN-101903347-A Piperidinyl and piperazinyl modulators of gamma-secretase JANSSEN PHARMACEUTICA NV 2010-12-01 CN disclosed