SCHEMBL28792136

SCHEMBL28792136

CCCCc1cc(N)n(CC)n1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.44
TLR7 Q9NYK1 4/20 0.43
ADORA2A P29274 3/20 0.40
ADORA2B P29275 3/20 0.40
CNR2 P34972 2/20 0.36
CNR1 P21554 1/20 0.36
HRH2 P25021 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
SKP2 Q13309 1/20 0.34
ALOX5 P09917 1/20 0.33
TLR8 Q9NR97 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
KCNH2 Q12809 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
IKBKB O14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27821973 0.87 NOS2 (0.43) NOS2TLR7ADORA2AADORA2BCNR2
SCHEMBL27836956 0.82 NOS2 (0.40) NOS2TLR7ADORA2AADORA2BCNR2
SCHEMBL7272832 0.81 NOS2 (0.44) NOS2TLR7ADORA2AADORA2BCNR2
SCHEMBL1292982 0.81 ADORA2A (0.40) ADORA2AADORA2B
SCHEMBL11070333 0.81 CNR2 (0.43) NOS2TLR7CNR2CNR1KCNH2
SCHEMBL28945481 0.80 NOS2 (0.38) NOS2TLR7CNR2KCNH2HRH4
SCHEMBL11691084 0.79 ADORA2A (0.45) NOS2ADORA2AADORA2BHRH3
SCHEMBL27841280 0.79 TLR7 (0.37) NOS2TLR7ADORA2AADORA2BCNR2
SCHEMBL27821985 0.77 TLR7 (0.36) NOS2TLR7ADORA2AADORA2BCNR2
SCHEMBL27841283 0.77 RAB9A (0.39) NOS2TLR7CNR2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105308046-A Kinase inhibitors CHIESI FARMA SPA 2016-02-03 CN disclosed
CN-102026985-A Quinazoline derivatives as RAF kinase modulators and methods and uses thereof AMBIT BIOSCIENCES CORPORATON 2011-04-20 CN disclosed