SCHEMBL28796115

SCHEMBL28796115

O=COC(c1ccccc1)N1CCNC(CO)C1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC6A4 P31645 5/20 0.36
ADRB1 P08588 1/20 0.36
OPRD1 P41143 7/20 0.35
SLC6A2 P23975 4/20 0.35
SLC6A3 Q01959 2/20 0.34
CACNA2D1 P54289 1/20 0.33
CACNA1B Q00975 1/20 0.33
CACNB1 Q02641 1/20 0.33
KCNH2 Q12809 2/20 0.33
CCR2 P41597 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28274309 0.82 HRH3 (0.38) MEN1KMT2ASLC6A4OPRD1SLC6A2
SCHEMBL27484196 0.79 MEN1 (0.54) MEN1KMT2ASLC6A4OPRD1SLC6A2
SCHEMBL28013093 0.78 HRH3 (0.43)
SCHEMBL27649776 0.77 KCNA3 (0.35)
SCHEMBL27838278 0.77 CYP2D6 (0.41) KCNH2
SCHEMBL27838235 0.76 LTA4H (0.37) MEN1KMT2ASLC6A4ADRB1SLC6A2
SCHEMBL27930040 0.73 KCNA3 (0.36) KMT2AKCNH2
Methane SCHEMBL28241933 0.73 KCNA3 (0.41) OPRD1OPRM1
SCHEMBL27625371 0.72 DPP4 (0.36) SLC6A2SLC6A3KCNH2OPRM1
SCHEMBL28762467 0.71 CYP2D6 (0.37) MEN1KMT2AOPRD1SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103030653-A Heteroarylopyrimidine derivative, medicinal salt thereof, methods for preparing heteroarylopyrimidine derivative and medicinal salt thereof and medical applications of heteroarylopyrimidine derivative and medicinal salt thereof SHANGHAI HENGRUI PHARM CO LTD 2013-04-10 CN disclosed
CN-102372706-A Phthalazinone derivative, its preparation method and application in medicament JIANGSU HENGRUI MEDICINE CO 2012-03-14 CN disclosed