SCHEMBL28797368

SCHEMBL28797368

CC(Br)c1cccc(C#N)c1F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.39
TSHR P16473 1/20 0.36
NOTUM Q6P988 1/20 0.35
ALDH1A1 P00352 4/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
LRRK2 Q5S007 1/20 0.32
AR P10275 1/20 0.32
EGLN2 Q96KS0 2/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
BCAT1 P54687 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
SOS1 Q07889 1/20 0.30
ANPEP P15144 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30762168 1.00 P2RX7 (0.39) P2RX7TSHRNOTUMALDH1A1L3MBTL1
SCHEMBL29278102 0.85 TSHR (0.34) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL9003991 0.85 GABRA1 (0.40) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL30762200 0.85 TSHR (0.34) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL24681944 0.81 CYP1A2 (0.40) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL16950500 0.81 NOTUM (0.38) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL31038398 0.81 CYP1A2 (0.40) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL30754463 0.81 CYP1A2 (0.40) TSHRNOTUMALDH1A1L3MBTL1LRRK2
SCHEMBL507010 0.80 TSHR (0.46) P2RX7TSHRALDH1A1L3MBTL1AR
SCHEMBL29974545 0.80 TSHR (0.46) P2RX7TSHRALDH1A1L3MBTL1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402081-A Aryl substituted amine derivative, preparation method and application thereof 南京医科大学 2024-01-16 CN disclosed
CN-103781775-A Metalloenzyme inhibitor compounds VIAMET PHARMACEUTICALS INC 2014-05-07 CN disclosed
CN-103380133-A Compounds and their use as BACE inhibitors ASTRAZENECA AB 2013-10-30 CN disclosed
CN-102459206-A Oxadiazole derivatives MERCK SERONO SA 2012-05-16 CN disclosed