SCHEMBL28797495

SCHEMBL28797495

O=C(O)N1Cc2cc(Br)ccc2C(c2ccc(F)cc2)C1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.52
ESR1 P03372 4/20 0.49
ESR2 Q92731 4/20 0.49
SLC6A2 P23975 6/20 0.47
SLC6A4 P31645 6/20 0.47
SLC6A3 Q01959 6/20 0.47
CYP2D6 P10635 1/20 0.47
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27869438 0.88 KIF11 (0.52) KIF11ESR1ESR2SLC6A2SLC6A4
SCHEMBL747351 0.83 KIF11 (0.48) KIF11ESR1ESR2SLC6A2SLC6A4
SCHEMBL752057 0.79 SLC6A2 (0.73) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL29104009 0.77 KIF11 (0.44) KIF11ESR1ESR2
SCHEMBL29238643 0.76 KIF11 (0.49) KIF11ESR1ESR2KMT2A
SCHEMBL22461557 0.76 KIF11 (0.55) KIF11ESR1ESR2SLC6A2SLC6A4
SCHEMBL22461558 0.76 KIF11 (0.55) KIF11ESR1ESR2SLC6A2SLC6A4
SCHEMBL751483 0.71 KIF11 (0.48) KIF11ESR1ESR2SLC6A2SLC6A4
SCHEMBL20533479 0.69 KIF11 (0.40) KIF11
SCHEMBL20533478 0.69 KIF11 (0.40) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102458123-A Aryl, heteroaryl, and heterocycle substituted tetrahydroisoquinolines and use thereof ALBANY MOLECULAR RES INC 2012-05-16 CN disclosed