SCHEMBL2880

SCHEMBL2880

CCOC(=O)c1c(-c2ccc(F)cc2)nc(N(NC)S(C)(=O)=O)nc1C(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.45
HMGCR P04035 2/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ALDH1A1 P00352 4/20 0.42
CYP3A4 P08684 1/20 0.42
PDE6D O43924 1/20 0.42
NR1I2 O75469 1/20 0.42
PDE4D Q08499 1/20 0.42
GCGR P47871 1/20 0.41
ABCC3 O15438 1/20 0.41
ABCC4 O15439 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3313 0.87 HMGCR (0.54) PTGS2HMGCRHDAC1HDAC2HDAC6
SCHEMBL3135 0.83 ALDH1A1 (0.45) PTGS2HMGCRHDAC1HDAC2HDAC6
SCHEMBL7922156 0.82 ALDH1A1 (0.43) PTGS2HMGCRALDH1A1CYP3A4PDE6D
SCHEMBL2768 0.81 PTGS2 (0.53) PTGS2ALDH1A1GCGRL3MBTL1NPC1
SCHEMBL15000315 0.80 HMGCR (0.52) PTGS2HMGCRHDAC1HDAC2HDAC6
SCHEMBL2211 0.79 ALDH1A1 (0.47) PTGS2ALDH1A1GCGRL3MBTL1NPC1
SCHEMBL13847948 0.79 ALDH1A1 (0.42) PTGS2HMGCRHDAC1HDAC2HDAC6
SCHEMBL15481445 0.79 ALDH1A1 (0.47) PTGS2ALDH1A1GCGRL3MBTL1NPC1
SCHEMBL13847940 0.78 ALDH1A1 (0.41) PTGS2HMGCRHDAC1HDAC2HDAC6
SCHEMBL1752130 0.78 HMGCR (0.56) HMGCRHDAC1HDAC2HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37314-E1 Pyrimidine derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 2001-08-07 US disclosed
US-5260440-A Anticholesterol agents SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed