SCHEMBL3135

SCHEMBL3135

CCOC(=O)c1c(-c2ccc(F)cc2)nc(N(C)S(=O)(=O)N(C)C)nc1C(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
HMGCR P04035 2/20 0.45
CYP3A4 P08684 1/20 0.45
PDE6D O43924 1/20 0.45
NR1I2 O75469 1/20 0.45
PDE4D Q08499 1/20 0.45
PTGS2 P35354 1/20 0.45
ABCC3 O15438 1/20 0.44
ABCC4 O15439 1/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
GCGR P47871 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3313 0.92 HMGCR (0.54) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL13847948 0.88 ALDH1A1 (0.42) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL7922156 0.86 ALDH1A1 (0.43) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL13847940 0.86 ALDH1A1 (0.41) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL13847937 0.85 ALDH1A1 (0.41) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL15000315 0.84 HMGCR (0.52) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL13847945 0.84 ALDH1A1 (0.40) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL2880 0.83 PTGS2 (0.45) ALDH1A1HMGCRCYP3A4PDE6DNR1I2
SCHEMBL15481445 0.81 ALDH1A1 (0.47) ALDH1A1PTGS2L3MBTL1GCGRKDM4E
SCHEMBL2768 0.81 PTGS2 (0.53) ALDH1A1PTGS2L3MBTL1GCGRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37314-E1 Pyrimidine derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 2001-08-07 US disclosed
US-5260440-A Anticholesterol agents SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
EP-0521471-A1 Pyrimidine derivatives as HMG-CoA reductase inhibitors SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-01-07 EP disclosed