SCHEMBL28801323

SCHEMBL28801323

Nc1c(-c2ccccc2)csc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.43
DAPK3 O43293 1/20 0.43
PRKD3 O94806 1/20 0.43
ABL1 P00519 1/20 0.43
NTRK1 P04629 1/20 0.43
LCK P06239 1/20 0.43
CSF1R P07333 1/20 0.43
RET P07949 1/20 0.43
MET P08581 1/20 0.43
PDGFRB P09619 1/20 0.43
FGFR1 P11362 1/20 0.43
PDGFRA P16234 1/20 0.43
PRKACA P17612 1/20 0.43
FLT1 P17948 1/20 0.43
LTK P29376 1/20 0.43
KDR P35968 1/20 0.43
MAP2K2 P36507 1/20 0.43
MAPK8 P45983 1/20 0.43
MAPK9 P45984 1/20 0.43
CSNK1A1 P48729 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151141 0.77 ALDH1A1 (0.51) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL29217099 0.74 DAPK3 (0.43) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL29217102 0.74 DAPK3 (0.43) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL7089546 0.72 KMT2A (0.48) ALDH1A1CYP2A6HSD17B10LMNASMN1; SMN2
SCHEMBL8219401 0.70 ALDH1A1 (0.49) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL3792808 0.69 ALDH1A1 (0.41) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL28687350 0.69 BTK (0.44) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL6271882 0.69 ALDH1A1 (0.54) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL15391338 0.69 PDPK1 (0.47) MAP4K4DAPK3PRKD3ABL1NTRK1
SCHEMBL8649337 0.68 CYP2A6 (0.60) ALDH1A1CYP2A6HSD17B10HPGDCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102970868-A Treatment of cancers having K-RAS mutations CURIS INC 2013-03-13 CN disclosed