SCHEMBL28801458

SCHEMBL28801458

Brc1cccc(-c2cc(Nc3cc[nH]c3)cs2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
MAPT P10636 1/20 0.35
HK1 P19367 1/20 0.35
RAB9A P51151 1/20 0.35
HKDC1 Q2TB90 1/20 0.35
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
CSNK2A1 P68400 1/20 0.34
CSNK2A3 Q8NEV1 1/20 0.34
CNR1 P21554 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B1 P14061 2/20 0.32
HSD17B2 P37059 2/20 0.32
SYK P43405 1/20 0.31
TYMP P19971 1/20 0.31
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27894484 0.87 MEN1 (0.33) ALDH1A1MAPTCNR1MEN1KMT2A
SCHEMBL27877864 0.84 HSD17B1 (0.36) MAPTCNR1MEN1KMT2AHSD17B1
SCHEMBL27877664 0.84 CNR1 (0.41) ALDH1A1MAPTRAB9ACNR1MEN1
SCHEMBL27877663 0.81 ESRRG (0.37) ALDH1A1HPGDMAPTHK1RAB9A
SCHEMBL27894480 0.79 CNR1 (0.44) ALDH1A1MAPTRAB9ACNR1MEN1
SCHEMBL8842433 0.76 RAPGEF4 (0.46) ALDH1A1MAPTMEN1KMT2AIDO1
SCHEMBL27894532 0.76 ACHE (0.37) ALDH1A1HPGDMAPTHK1RAB9A
SCHEMBL27894478 0.75 KMT2A (0.53) ALDH1A1HPGDMAPTRAB9AMEN1
SCHEMBL28137854 0.67 IDO1 (0.42) ALDH1A1HPGDMAPTRAB9AMEN1
SCHEMBL27894479 0.67 MEN1 (0.35) ALDH1A1MAPTCNR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104628741-A Novel compounds and therapeutic use thereof for protein kinase inhibition WU ZHANGGUI 2015-05-20 CN claimed
CN-102711475-B Novel compounds and their therapeutic use for inhibiting protein kinases WU ZHANGGUI 2015-01-28 CN claimed
CN-102711475-A Novel compounds and their therapeutic use for inhibiting protein kinases ZHANGGUI WU 2012-10-03 CN claimed
CN-104628741-A Novel compounds and therapeutic use thereof for protein kinase inhibition WU ZHANGGUI 2015-05-20 CN disclosed
CN-102711475-B Novel compounds and their therapeutic use for inhibiting protein kinases WU ZHANGGUI 2015-01-28 CN disclosed