SCHEMBL28801601

SCHEMBL28801601

O=C1CCN1Cc1ccc(F)cc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
POLB P06746 1/20 0.61
RAB9A P51151 1/20 0.56
L3MBTL1 Q9Y468 4/20 0.54
HTT P42858 3/20 0.54
HRH3 Q9Y5N1 1/20 0.50
LMNA P02545 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
TP53 P04637 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.46
NPC1 O15118 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GRM2 Q14416 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5578262 0.89 L3MBTL1 (0.65) ALDH1A1POLBRAB9AL3MBTL1HTT
SCHEMBL4501555 0.89 L3MBTL1 (0.70) ALDH1A1POLBRAB9AL3MBTL1HTT
SCHEMBL1534180 0.86 ALDH1A1 (0.54) ALDH1A1POLBRAB9AL3MBTL1HTT
SCHEMBL7389188 0.80 L3MBTL1 (0.73) POLBRAB9AL3MBTL1HRH3NPC1
SCHEMBL2899901 0.79 ALDH1A1 (0.63) ALDH1A1POLBRAB9AL3MBTL1HTT
SCHEMBL11200681 0.78 L3MBTL1 (0.76) L3MBTL1HRH3SMN1; SMN2KMT2A
SCHEMBL15858005 0.78 ALDH1A1 (0.53) ALDH1A1POLBRAB9AL3MBTL1HTT
SCHEMBL8325711 0.78 GRM2 (0.54) ALDH1A1POLBRAB9AL3MBTL1HTT
SCHEMBL2203678 0.78 ALDH1A1 (0.53) ALDH1A1POLBRAB9AL3MBTL1HTT
Hydrochloric Acid SCHEMBL4767938 0.78 ALDH1A1 (0.61) ALDH1A1POLBRAB9AL3MBTL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958922-B 2,5,6,7-tetrahydrochysene-[Isosorbide-5-Nitrae] oxygen azepine *-3-base amine or 2,3,6,7-tetrahydrochysene-[Isosorbide-5-Nitrae] oxygen azepine *-5-ylamine compounds HOFFMAN-LA ROCHE LTD. (CH) 2015-09-30 CN disclosed
CN-102958922-A 2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine or 2,3,6,7-tetrahydro-[1,4]oxazepin-5-ylamine compounds HOFFMANN LA ROCHE 2013-03-06 CN disclosed