SCHEMBL5578262

SCHEMBL5578262

O=C1CCCN1Cc1ccc(F)cc1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.65
HRH3 Q9Y5N1 1/20 0.59
ALDH1A1 P00352 2/20 0.57
POLB P06746 1/20 0.57
ACACB O00763 1/20 0.54
RAB9A P51151 1/20 0.53
GRM2 Q14416 3/20 0.52
HTT P42858 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
GRIA2 P42262 1/20 0.50
MAPT P10636 1/20 0.48
RECQL P46063 1/20 0.48
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4501555 0.96 L3MBTL1 (0.70) L3MBTL1HRH3ALDH1A1POLBACACB
SCHEMBL11200681 0.91 L3MBTL1 (0.76) L3MBTL1HRH3ACACBKMT2ACYP1A2
SCHEMBL28801601 0.89 ALDH1A1 (0.61) L3MBTL1HRH3ALDH1A1POLBRAB9A
SCHEMBL19717008 0.84 L3MBTL1 (0.67) L3MBTL1HRH3ACACBKMT2ACYP1A2
SCHEMBL10399987 0.84 L3MBTL1 (0.67) L3MBTL1HRH3ALDH1A1ACACBRAB9A
SCHEMBL3903106 0.82 L3MBTL1 (0.65) L3MBTL1HRH3ACACBKMT2ACYP1A2
SCHEMBL6824717 0.82 L3MBTL1 (0.65) L3MBTL1HRH3POLBACACBKMT2A
SCHEMBL256037 0.82 L3MBTL1 (0.65) L3MBTL1HRH3ACACBKMT2ACYP1A2
SCHEMBL13853398 0.82 L3MBTL1 (0.65) L3MBTL1HRH3ACACBGRM2HTT
SCHEMBL13215733 0.82 L3MBTL1 (0.65) L3MBTL1HRH3ALDH1A1ACACBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4127157-B1 MODIFIED DIPEPTIDE CLEAVASES, USES THEREOF AND RELATED KITS ENCODIA INC (US) 2026-02-11 EP claimed
WO-2025060978-A1 TRICYCLIC PYRIDINE COMPOUND ACTING AS SARM1 ENZYME ACTIVITY INHIBITOR, AND USE THEREOF 科辉智药(深圳)新药研究中心有限公司 2025-03-27 WO disclosed
CN-117916241-A Spiro compounds 阿斯利康(瑞典)有限公司 2024-04-19 CN disclosed
EP-3292101-B1 TRICYCLIC SULFONES AS ROR-GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2021-07-28 EP disclosed
EP-3362441-B1 SELECTIVE NR2B ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2020-08-12 EP disclosed
WO-2017066366-A1 SELECTIVE NR2B ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-04-20 WO disclosed
EP-3092224-A1 SELECTIVE NR2B ANTAGONISTS Bristol-Myers Squibb Company (US) 2016-11-16 EP disclosed
WO-2015105772-A1 SELECTIVE NR2B ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-07-16 WO disclosed
US-20070232538-A1 Uses of polypeptides TAKEDA PHARMACEUTICAL COMPANY, LTD (JP) 2007-10-04 US disclosed
US-20040053826-A1 Uses of polypeptides TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-03-18 US disclosed
US-20030139442-A1 Vasoactive agents TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2003-07-24 US disclosed
EP-1308513-A1 USE OF POLYPEPTIDE Takeda Chemical Industries, Ltd. (JP) 2003-05-07 EP disclosed
EP-1262195-A1 VASOACTIVE AGENTS Takeda Chemical Industries, Ltd. (JP) 2002-12-04 EP disclosed
US-4189495-A TREATMENT OF NERVOUS AND PSYCHOSOMATIC DISORDERS SYNTHELABO (FR) 1980-02-19 US disclosed
US-4172143-A PSYCHOSOMATIC AND PSYCHOLOGICAL DISTURBANCES SYNTHELABO (FR) 1979-10-23 US disclosed
US-4158060-A PSYCHOLOGICAL DISORDERS SYNTHELABO (FR) 1979-06-12 US disclosed
US-4021567-A FOR PSYCHOSOMATIC AND PSYCHOTIC DISTURBANCES SYNTHELABO (FR) 1977-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030139442-A1 Vasoactive agents VIPR2, VIPR1, GPR4 L3MBTL1 4672/4885HRH3 512/4885ALDH1A1 2435/4885
US-20070232538-A1 Uses of polypeptides NPSR1, SCTR, GRPR L3MBTL1 3149/4885HRH3 202/4885ALDH1A1 3946/4885
US-20040053826-A1 Uses of polypeptides NPSR1, SCTR, GRPR L3MBTL1 3149/4885HRH3 202/4885ALDH1A1 3946/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.