SCHEMBL28802185

SCHEMBL28802185

Cc1ccc(N)c(-c2ccccc2)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.44
ALDH1A1 P00352 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
TSHR P16473 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPK1 P28482 2/20 0.44
CASP3 P42574 1/20 0.44
HBB P68871 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CD44 P16070 1/20 0.43
KMT2A Q03164 3/20 0.41
BRD4 O60885 1/20 0.41
TDO2 P48775 1/20 0.41
AKT2 P31751 1/20 0.41
MAPT P10636 3/20 0.40
CDK8 P49336 1/20 0.40
ACVR1 Q04771 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8321808 0.86 KMT2A (0.44) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL3794847 0.84 CYP3A4 (0.46) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL28726060 0.83 ALDH1A1 (0.43) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL4447138 0.83 KMT2A (0.41) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL614879 0.81 ALDH1A1 (0.44) CYP3A4ALDH1A1SMN1; SMN2TSHRMAPK1
SCHEMBL29799881 0.81 ALDH1A1 (0.44) CYP3A4ALDH1A1SMN1; SMN2TSHRMAPK1
SCHEMBL27685032 0.81 NPC1 (0.52) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL28155065 0.79 MAPT (0.42) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL27397239 0.79 SMN1; SMN2 (0.44) CYP3A4ALDH1A1SMN1; SMN2TSHRNPC1
SCHEMBL25014 0.78 HSD17B10 (0.50) CYP3A4ALDH1A1SMN1; SMN2TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107148420-A Benzyl substituted indazoles 拜耳制药股份公司 2017-09-08 CN disclosed
CN-107074825-A Benzyl substituted indazoles as BUB1 kinase inhibitors 拜耳制药股份公司 2017-08-18 CN disclosed
CN-102791659-A Material for electronic devices MERCK PATENT GMBH 2012-11-21 CN disclosed