SCHEMBL28806402

SCHEMBL28806402

COc1ccc(-c2cccc(Cl)c2Cl)s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.42
NUDT1 P36639 1/20 0.35
SLC6A3 Q01959 1/20 0.35
P2RX7 Q99572 3/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
SLC16A3 O15427 1/20 0.33
SLC16A1 P53985 1/20 0.33
MCTS1 Q9ULC4 1/20 0.33
NOTUM Q6P988 1/20 0.33
IDO1 P14902 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28804554 0.86 APP (0.48) APPKMT2AALDH1A1MAPTHPGD
SCHEMBL2407370 0.78 TSHR (0.39) SLC6A3KMT2AHPGDTUBB4ATUBB
SCHEMBL6927360 0.73 SLC6A3 (0.48) SLC6A3KMT2AALDH1A1MAPTHPGD
SCHEMBL14871942 0.70 APP (0.46) APPPDGFRBPDGFRATUBB4ATUBB
SCHEMBL3960432 0.70 APP (0.48) APPKMT2AALDH1A1HPGDPDGFRB
SCHEMBL1727532 0.69 CYP2E1 (0.46) APPKMT2AALDH1A1MAPTHPGD
SCHEMBL2413548 0.69 AVPR2 (0.38) P2RX7NOTUMIDO1TSHRCYP2D6
SCHEMBL2407673 0.69 CYP2A6 (0.46) P2RX7KMT2AALDH1A1MAPTHPGD
SCHEMBL2407368 0.68 HPGD (0.61) KMT2AALDH1A1HPGDTSHR
SCHEMBL440943 0.67 TSHR (0.52) NUDT1P2RX7NOTUMIDO1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103189363-B Biaryl linked aryl triazolones and uses thereof BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-29 CN disclosed
CN-103189363-A Biaryl linked aryl triazolones and uses thereof BAYER IP GMBH 2013-07-03 CN disclosed