SCHEMBL28809051

SCHEMBL28809051

O=C(C=Cc1ccc(-c2ccccc2)cc1)Nc1ccccc1C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM2 O94759 6/20 1.00
LTB4R Q15722 3/20 1.00
TRPA1 O75762 7/20 0.77
TRPM8 Q7Z2W7 4/20 0.77
MEN1 O00255 4/20 0.71
KMT2A Q03164 4/20 0.71
NPC1 O15118 3/20 0.71
RAB9A P51151 3/20 0.71
SMN1; SMN2 Q16637 3/20 0.71
MAPT P10636 2/20 0.71
PLA2G1B P04054 1/20 0.64
CYSLTR2 Q9NS75 1/20 0.64
CYSLTR1 Q9Y271 1/20 0.64
ALDH1A1 P00352 2/20 0.63
TP53 P04637 2/20 0.63
CYP3A4 P08684 2/20 0.63
HPGD P15428 2/20 0.63
HIF1A Q16665 2/20 0.63
KDM4E B2RXH2 2/20 0.63
APEX1 P27695 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28809046 1.00 TRPM2 (1.00) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL294403 0.91 TRPM2 (0.83) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL294402 0.91 TRPM2 (0.83) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL2778922 0.90 TRPM2 (0.81) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL2778920 0.90 TRPM2 (0.81) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL29401064 0.90 TRPM2 (0.81) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL2781343 0.87 MEN1 (0.78) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL2779999 0.87 TRPA1 (1.00) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL2779997 0.87 TRPA1 (1.00) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL2781340 0.87 MEN1 (0.78) TRPM2LTB4RTRPA1TRPM8MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114831977-A Application of benzoic acid derivatives as TRPM2 protein inhibitors 北京大学 2022-08-02 CN claimed
CN-114831977-B Application of benzoic acid derivative as TRPM2 protein inhibitor 北京大学 2023-12-19 CN disclosed
CN-114831977-A Application of benzoic acid derivatives as TRPM2 protein inhibitors 北京大学 2022-08-02 CN disclosed