SCHEMBL28809073

SCHEMBL28809073

COC(=O)c1c(C(F)(F)F)ccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 1/20 0.54
KCNJ11 Q14654 11/20 0.47
ABCC9 O60706 6/20 0.47
ABCC8 Q09428 6/20 0.47
KCNJ8 Q15842 6/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 1/20 0.46
NOTUM Q6P988 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
RCE1 Q9Y256 1/20 0.43
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
NR4A2 P43354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3370877 0.80 HPGD (0.53) KCNJ11ABCC9ABCC8KCNJ8MEN1
SCHEMBL10587314 0.79 KDM4E (0.46) KCNJ11ABCC9ABCC8KCNJ8MEN1
SCHEMBL15414915 0.79 NCEH1 (0.58) NCEH1MEN1KMT2AKDM4EALDH1A1
SCHEMBL1994212 0.78 CA12 (0.55) KDM4ENOTUMALDH1A1HPGDLMNA
SCHEMBL14052468 0.77 BACE1 (0.47) NCEH1KCNJ11TRPV1LMNAMAPK1
SCHEMBL12985269 0.77 KCNJ11 (0.42) NCEH1KCNJ11ABCC9ABCC8KCNJ8
SCHEMBL1638703 0.77 CA12 (0.60) NCEH1MEN1KMT2AKDM4EALDH1A1
SCHEMBL71131 0.77 NCEH1 (0.59) NCEH1MEN1KMT2AKDM4EALDH1A1
SCHEMBL29404644 0.77 NCEH1 (0.59) NCEH1MEN1KMT2AKDM4EALDH1A1
SCHEMBL1648076 0.77 NCEH1 (0.59) NCEH1MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103443099-A Compositions and methods for modulating FXR IRM LLC 2013-12-11 CN disclosed
CN-103370315-A Compositions and methods for modulating farnesoid x receptors IRM LLC 2013-10-23 CN disclosed