SCHEMBL28809104

SCHEMBL28809104

Fc1ccc(-c2ccnn2-c2ccccc2N2CCOCC2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.46
KDM4A O75164 1/20 0.46
KDM5A P29375 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
KDM5B Q9UGL1 1/20 0.46
HSP90AA1 P07900 1/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
P2RX7 Q99572 1/20 0.40
AR P10275 1/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 2/20 0.39
ATR Q13535 1/20 0.39
ATRIP Q8WXE1 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALOX15 P16050 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27933174 0.88 HSP90AA1 (0.45) LRRK2HSP90AA1MEN1KMT2AAR
SCHEMBL28809098 0.85 KDM4A (0.47) LRRK2KDM4AKDM5AKDM4CKDM5B
SCHEMBL28807011 0.83 ALDH1A1 (0.48) LRRK2KDM5AKDM4CKDM5BKMT2A
SCHEMBL27948412 0.82 KDM5A (0.46) LRRK2KDM5AKDM4CKDM5BMEN1
SCHEMBL27948410 0.81 HPGD (0.48) HSP90AA1MEN1KMT2AP2RX7ALDH1A1
SCHEMBL27948419 0.80 NR3C2 (0.43) KDM5AKDM4CKDM5BHSP90AA1MEN1
SCHEMBL27933075 0.78 CNR2 (0.51) LRRK2MEN1KMT2AALDH1A1HPGD
SCHEMBL27932732 0.77 PTGS2 (0.50) ARALDH1A1HSD17B10SMN1; SMN2NPSR1
SCHEMBL28903748 0.75 MAP4K1 (0.49) LRRK2MEN1KMT2AALDH1A1HPGD
SCHEMBL27932740 0.75 MAPK9 (0.47) MEN1KMT2AARHSD17B10ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103492389-A Pyrazolo [4, 3-d] pyrimidines useful as kinase inhibitors ORIGENIS GMBH 2014-01-01 CN claimed
CN-103492389-A Pyrazolo [4, 3-d] pyrimidines useful as kinase inhibitors ORIGENIS GMBH 2014-01-01 CN disclosed