SCHEMBL28809348

SCHEMBL28809348

O=C(Nc1cccc(Br)n1)c1c(F)cc(F)cc1F

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
HTR1F P30939 6/20 0.54
CHRM5 P08912 1/20 0.54
DRD5 P21918 1/20 0.54
HTR1D P28221 1/20 0.54
HTR1E P28566 1/20 0.54
HTR7 P34969 1/20 0.54
OPRK1 P41145 1/20 0.54
TMEM97 Q5BJF2 1/20 0.54
SIGMAR1 Q99720 1/20 0.54
HTR1A P08908 1/20 0.54
HTR1B P28222 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54
GRM5 P41594 4/20 0.49
NPC1 O15118 1/20 0.47
CYP1A2 P05177 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16321125 0.89 MEN1 (0.78) MEN1KMT2AGRM5NPC1CYP1A2
SCHEMBL28808156 0.83 HTR1F (0.56) MEN1KMT2AHTR1FGRM5NPC1
SCHEMBL1196838 0.82 MEN1 (0.62) MEN1KMT2AHTR1FCHRM5DRD5
SCHEMBL23733271 0.82 GRM5 (0.72) MEN1KMT2AHTR1FCHRM5DRD5
SCHEMBL23733275 0.82 MEN1 (0.62) MEN1KMT2AHTR1FCHRM5DRD5
SCHEMBL23733250 0.80 HTR1F (0.61) MEN1KMT2AHTR1FCHRM5DRD5
SCHEMBL23702725 0.79 HTR1F (0.60) MEN1KMT2AHTR1FCHRM5DRD5
SCHEMBL28808130 0.79 CHRNB2 (0.60) MEN1KMT2AHTR1FGRM5NPC1
SCHEMBL31052662 0.78 KMT2A (0.56) MEN1KMT2AHTR1FCHRM5DRD5
SCHEMBL23702723 0.78 HTR1F (0.58) MEN1KMT2AHTR1FCHRM5DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113045540-B Preparation method of masmipide 上海天慈国际药业有限公司 2024-02-13 CN claimed
CN-113045540-A Preparation method of rasemiptan 上海天慈国际药业有限公司 2021-06-29 CN claimed
CN-113045540-B Preparation method of masmipide 上海天慈国际药业有限公司 2024-02-13 CN disclosed
CN-114728929-A Pyridine methylene piperidine derivatives and use thereof 广东东阳光药业有限公司 2022-07-08 CN disclosed
CN-113045540-A Preparation method of rasemiptan 上海天慈国际药业有限公司 2021-06-29 CN disclosed