SCHEMBL28809379

SCHEMBL28809379

CCn1c2ccccc2c2cc(/C=C\C(=O)O)c(C#N)cc21

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.48
KDM4E B2RXH2 6/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 2/20 0.45
MAPK1 P28482 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
DHODH Q02127 1/20 0.45
MAPT P10636 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HPGD P15428 1/20 0.45
CASP1 P29466 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PKM P14618 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28810410 0.86 DHODH (0.52) RORCKDM4ELMNAPOLBMAPK1
SCHEMBL28809982 0.85 KDM4E (0.47) KDM4EMAPTALDH1A1HPGDHSD17B10
SCHEMBL13170473 0.79 KDM4E (0.61) KDM4ELMNAPOLBMAPK1NPSR1
SCHEMBL13170385 0.79 KDM4E (0.61) KDM4ELMNAPOLBMAPK1NPSR1
SCHEMBL4631887 0.75 KDM4E (0.56) RORCKDM4ELMNAPOLBMAPK1
SCHEMBL4631890 0.75 KDM4E (0.56) RORCKDM4ELMNAPOLBMAPK1
SCHEMBL28811113 0.75 MAPT (0.45) KDM4ELMNAMAPK1NPSR1DHODH
SCHEMBL8964807 0.74 TP53 (0.49) RORCKDM4ELMNAPOLBMAPK1
SCHEMBL27619336 0.72 KDM4E (0.55) KDM4ELMNAPOLBMAPK1NPSR1
SCHEMBL8921074 0.71 KDM4E (0.53) KDM4ELMNAPOLBMAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109970622-B 2-substituent-3- (9-alkyl-9H-carbazole-3-yl) acrylonitrile compound and preparation method thereof 陕西科技大学 2022-06-07 CN disclosed