SCHEMBL28810071

SCHEMBL28810071

O=C(/C=C/c1ccc(-c2ccccc2)cc1C(F)(F)F)Nc1ccccc1C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM2 O94759 5/20 0.67
LTB4R Q15722 1/20 0.62
TRPA1 O75762 7/20 0.58
TRPM8 Q7Z2W7 4/20 0.58
MAOB P27338 2/20 0.51
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KDM4E B2RXH2 2/20 0.48
APEX1 P27695 2/20 0.48
MAPT P10636 2/20 0.48
POLB P06746 1/20 0.48
RECQL P46063 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAOA P21397 1/20 0.48
ALDH1A1 P00352 2/20 0.47
TP53 P04637 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28810074 1.00 TRPM2 (0.67) TRPM2LTB4RTRPA1TRPM8MAOB
SCHEMBL8048012 0.86 MAOB (0.69) TRPM2LTB4RTRPA1TRPM8MAOB
SCHEMBL8048008 0.86 MAOB (0.69) TRPM2LTB4RTRPA1TRPM8MAOB
SCHEMBL28810087 0.85 TRPM2 (0.68) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL28810088 0.85 TRPM2 (0.68) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL28810093 0.82 TRPM2 (0.67) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL28808953 0.82 TRPM2 (0.67) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL28809601 0.82 TRPA1 (0.73) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL28809597 0.82 TRPA1 (0.73) TRPM2LTB4RTRPA1TRPM8MEN1
SCHEMBL28808950 0.82 TRPM2 (0.67) TRPM2LTB4RTRPA1TRPM8MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114831977-A Application of benzoic acid derivatives as TRPM2 protein inhibitors 北京大学 2022-08-02 CN claimed
CN-114831977-B Application of benzoic acid derivative as TRPM2 protein inhibitor 北京大学 2023-12-19 CN disclosed
CN-114831977-A Application of benzoic acid derivatives as TRPM2 protein inhibitors 北京大学 2022-08-02 CN disclosed