SCHEMBL2881114

SCHEMBL2881114

CCN(CC)Cc1ccc(CCn2ccc(OCc3ccccc3)nc2=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 11/20 0.57
L3MBTL1 Q9Y468 1/20 0.46
BCHE P06276 6/20 0.43
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5265127 0.75 MAPK14 (0.58) PKM
SCHEMBL5266116 0.72 GRM5 (0.44) MCHR1PKM
SCHEMBL2881979 0.72 MCHR1 (1.00) MCHR1
SCHEMBL2883772 0.70 MCHR1 (0.56) MCHR1BCHE
SCHEMBL19746414 0.70 P2RX7 (0.46) MCHR1L3MBTL1
SCHEMBL17554285 0.70 EP300 (0.44) MCHR1L3MBTL1
SCHEMBL4002396 0.68 MCHR1 (0.82) MCHR1
SCHEMBL1366606 0.68 MCHR1 (0.47) MCHR1PKM
SCHEMBL2884206 0.68 MCHR1 (1.00) MCHR1BCHE
SCHEMBL1364736 0.66 MCHR1 (0.73) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100216758-A1 Pyridone Compounds MSD K.K. (JP) 2010-08-26 US disclosed
EP-1916239-A1 PYRIDONE COMPOUND BANYU PHARMACEUTICAL CO., LTD. (JP) 2008-04-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100216758-A1 Pyridone Compounds NPY1R, MC5R, MC1R MCHR1 4/4885L3MBTL1 979/4885BCHE 2805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.