SCHEMBL28811371

SCHEMBL28811371

Cc1c(C(=O)O)cccc1C(=O)O.c1nc2c3cc-3cc2s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.48
SLC22A12 Q96S37 1/20 0.48
SYK P43405 2/20 0.38
KDM4E B2RXH2 7/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
TSHR P16473 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HKDC1 Q2TB90 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 4/20 0.36
USP2 O75604 1/20 0.36
PTGER1 P34995 1/20 0.35
MYC P01106 1/20 0.35
LDHA P00338 1/20 0.35
HSD17B10 Q99714 2/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982298 0.73 KDM4E (0.42) XDHSLC22A12KDM4ENPC1RAB9A
SCHEMBL262049 0.73 ALDH1A1 (0.44) XDHSLC22A12KDM4ENPC1RAB9A
Benzene SCHEMBL27265959 0.70 TSHR (0.61) KDM4ENPC1RAB9ATSHRL3MBTL1
SCHEMBL27703149 0.70 TSHR (0.61) KDM4ENPC1RAB9ATSHRL3MBTL1
SCHEMBL756585 0.70 TSHR (0.61) KDM4ENPC1RAB9ATSHRL3MBTL1
SCHEMBL27786189 0.69 ACMSD (0.53) KDM4ENPC1RAB9ATSHRTDP1
SCHEMBL10768142 0.68 TSHR (0.59) KDM4ENPC1RAB9ATSHRL3MBTL1
Fluoride SCHEMBL27323288 0.68 TSHR (0.59) KDM4ENPC1RAB9ATSHRL3MBTL1
Water SCHEMBL27479836 0.68 TSHR (0.59) KDM4ENPC1RAB9ATSHRL3MBTL1
Ethane SCHEMBL27288094 0.68 TSHR (0.59) KDM4ENPC1RAB9ATSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103880827-B The application of the reuptake of aryl and the substituted tetrahydroisoquinoline of heteroaryl and blocking-up norepinephrine, dopamine and serotonin 阿尔巴尼分子研究公司 2017-01-04 CN disclosed
CN-103880827-A Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin ALBANY MOLECULAR RES INC 2014-06-25 CN disclosed