SCHEMBL28813367

SCHEMBL28813367

CC(=O)Oc1cc(C(C)c2ccccc2)sc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 2/20 0.40
TSHR P16473 2/20 0.40
HPGD P15428 2/20 0.40
ESR1 P03372 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
HMGB1 P09429 1/20 0.40
GGT1 P19440 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
BLM P54132 1/20 0.40
NAPRT Q6XQN6 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTT P42858 1/20 0.38
KMT2A Q03164 2/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP1A2 P05177 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27965937 0.82 TNFSF11 (0.37) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL5099235 0.75 IKBKB (0.53) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL14875542 0.75 ALDH1A1 (0.58) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL27712944 0.74 MAPT (0.56) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL28813368 0.73 ADORA2A (0.38) HPGDPTGS1PTGS2KMT2ACYP1A2
SCHEMBL868867 0.72 PTGS2 (0.53) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL27785358 0.69 PTGS2 (0.48) KDM4EALDH1A1HSD17B10TSHRHPGD
Trifluoroacetic Acid SCHEMBL5092977 0.69 IKBKB (0.46) ALDH1A1HPGDKMT2AMAPTCYP1A2
SCHEMBL27789075 0.69 ALDH1A1 (0.45) KDM4EALDH1A1HSD17B10TSHRHPGD
SCHEMBL7886963 0.69 NPC1 (0.47) ALDH1A1KMT2AMAPTMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103958521-A Pyrimidin-4-one derivatives and their use in the treatment, alleviation or prevention of viral diseases HOFFMANN LA ROCHE 2014-07-30 CN disclosed
CN-103958475-A Heteroaryl hydroxamic acid derivatives and their use in the treatment, alleviation or prevention of viral diseases HOFFMANN LA ROCHE 2014-07-30 CN disclosed