SCHEMBL28816404

SCHEMBL28816404

COc1cc(N)c(CC2CCN(CC(O)COc3cccc(Cl)c3Cl)CC2)cc1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.47
DRD4 P21917 6/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ATM Q13315 1/20 0.46
DRD2 P14416 1/20 0.45
GAA P10253 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
USP2 O75604 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997566 0.94 MEN1 (0.51) ABCB1DRD4MEN1KMT2AATM
SCHEMBL27997734 0.92 ABCB1 (0.45) ABCB1DRD4MEN1KMT2AATM
SCHEMBL27997518 0.88 ALDH1A1 (0.46) ABCB1DRD4MEN1KMT2AATM
SCHEMBL27997735 0.86 HRH1 (0.48) ABCB1DRD4MEN1KMT2AATM
SCHEMBL27997716 0.86 DRD4 (0.55) DRD4MEN1KMT2AGAALMNA
SCHEMBL27997713 0.86 DRD4 (0.56) ABCB1DRD4MEN1KMT2ADRD2
SCHEMBL27997731 0.84 TSHR (0.52) ABCB1DRD4MEN1KMT2AGAA
SCHEMBL27997717 0.83 DRD4 (0.51) ABCB1DRD4MEN1KMT2AGAA
SCHEMBL27997565 0.82 ACHE (0.46) DRD4MEN1KMT2ADRD2ADRB2
SCHEMBL2331564 0.82 HTR4 (0.62) DRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102186840-B Piperidine compounds, pharmaceutical compositions containing the same and uses thereof SK BIOPHARMACEUTICALS CO LTD 2015-03-25 CN disclosed