SCHEMBL28816713

SCHEMBL28816713

CC(ONC(=O)c1ccccc1)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 2/20 0.47
POLB P06746 1/20 0.47
KDM4E B2RXH2 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
RAB9A P51151 8/20 0.44
NPC1 O15118 7/20 0.44
HPGD P15428 1/20 0.43
MLYCD O95822 1/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HDAC3 O15379 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
IDO1 P14902 1/20 0.41
ALOX15 P16050 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27480093 0.81 ALDH1A1 (0.52) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL5390967 0.80 ALDH1A1 (0.55) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL28124499 0.77 ALDH1A1 (0.52) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL1695124 0.77 ALDH1A1 (0.55) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL28306142 0.76 ALDH1A1 (0.50) ALDH1A1KMT2AMAPTPOLBKDM4E
Benzoic Acid Hydrazide SCHEMBL10824591 0.75 ALDH1A1 (0.45) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL6291224 0.75 RAB9A (0.49) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL11143477 0.75 RAB9A (0.55) ALDH1A1KMT2AMAPTPOLBKDM4E
SCHEMBL28884941 0.74 KMT2A (0.54) ALDH1A1KMT2AMAPTPOLBTDP1
SCHEMBL30771879 0.74 SMN1; SMN2 (0.50) ALDH1A1KMT2ARAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114630822-A Biaryl dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-06-14 CN disclosed
CN-114286813-A Substituted urea dihydroorotate dehydrogenase inhibitors 詹森生物科技公司 2022-04-05 CN disclosed