SCHEMBL28817028

SCHEMBL28817028

N=C(N)c1cnc(F)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.40
UBE2T Q9NPD8 2/20 0.36
F2 P00734 3/20 0.36
F10 P00742 2/20 0.36
PRSS1 P07477 3/20 0.35
PRSS2 P07478 3/20 0.35
PRSS3 P35030 3/20 0.35
C1S P09871 1/20 0.35
F12 P00748 1/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
PKM P14618 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
PRMT1 Q99873 1/20 0.33
LMNA P02545 1/20 0.32
BLM P54132 1/20 0.32
MASP2 O00187 1/20 0.32
PLAU P00749 1/20 0.32
THPO P40225 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1828070 0.79 NNMT (0.44) BACE1LMNA
SCHEMBL30445761 0.79 NNMT (0.44) BACE1LMNA
SCHEMBL30936080 0.77 F10 (0.33) UBE2TF2F10PRSS1PRSS2
SCHEMBL30721127 0.72 HCAR2 (0.50) LMNA
SCHEMBL898595 0.72 HCAR2 (0.50) LMNA
SCHEMBL20577332 0.71 BACE1 (0.33) BACE1
SCHEMBL12634680 0.70 CES2 (0.50) F2F10PRSS1PRSS2PRSS3
Hydrochloric Acid SCHEMBL5115579 0.69 CES2 (0.48) F2F10PRSS1PRSS2PRSS3
SCHEMBL20554192 0.68 UBE2T (0.49) UBE2TF2F10PRSS1PRSS3
SCHEMBL8005179 0.68 HCAR2 (0.55) F2F10PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104302626-A 4, 4-disubstituted-1, 4-dihydropyrimidines and their use as medicaments for the treatment of hepatitis b JANSSEN R & D IRELAND 2015-01-21 CN disclosed