SCHEMBL28819645

SCHEMBL28819645

COc1ccc(-c2nc3cc(F)c(F)cc3n2C(C(N)=O)(C2CCCCC2)C2CCCCC2)c(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.42
POLB P06746 2/20 0.40
HTT P42858 1/20 0.38
HSP90AA1 P07900 1/20 0.38
NR1H4 Q96RI1 3/20 0.38
TP53 P04637 1/20 0.38
PIK3CA P42336 1/20 0.38
DHODH Q02127 1/20 0.37
PLAU P00749 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX5AP P20292 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ATM Q13315 1/20 0.35
DPP4 P27487 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819691 0.90 ADORA3 (0.41) ADORA3POLBHTTHSP90AA1NR1H4
SCHEMBL28819665 0.89 POLB (0.40) ADORA3POLBHTTNR1H4TP53
SCHEMBL28819544 0.88 POLB (0.41) ADORA3POLBHTTNR1H4TP53
Hydrochloric Acid SCHEMBL4209518 0.88 POLB (0.40) ADORA3POLBHTTTP53PLAU
SCHEMBL28819518 0.87 POLB (0.47) ADORA3POLBHSP90AA1TP53PLAU
Hydrochloric Acid SCHEMBL4209516 0.87 POLB (0.40) ADORA3POLBHTTTP53PLAU
SCHEMBL28819643 0.82 POLB (0.40) ADORA3POLBHTTTP53PLAU
SCHEMBL28819618 0.80 TP53 (0.44) POLBTP53KDM4EALDH1A1
SCHEMBL28819648 0.79 NR1H4 (0.45) NR1H4KMT2AALDH1A1CYP11B1CYP11B2
SCHEMBL28819577 0.79 CNR2 (0.43) POLBTP53KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110404073-B Methods and pharmaceutical compositions for treating hepatitis B virus infection 国家医疗保健研究所 2022-08-16 CN disclosed