SCHEMBL28822256

SCHEMBL28822256

Clc1ccc(Oc2ccc(-c3cc[nH]n3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 6/20 0.51
HAO1 Q9UJM8 2/20 0.51
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
METAP2 P50579 1/20 0.43
NOTUM Q6P988 1/20 0.43
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PTGS2 P35354 1/20 0.40
SLC2A1 P11166 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
CDH1 P12830 1/20 0.39
CTNNB1 P35222 1/20 0.39
TCF7L2 Q9NQB0 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1645103 0.90 METAP2 (0.50) LTA4HHAO1METAP2NOTUMMAPT
Hydrochloric Acid SCHEMBL10565482 0.88 METAP2 (0.48) LTA4HHAO1METAP2NOTUMMAPT
Methylamine SCHEMBL27885520 0.85 METAP2 (0.46) LTA4HHAO1METAP2NOTUMMAPT
SCHEMBL3364770 0.83 NPC1 (0.50) LTA4HHAO1MAOA
SCHEMBL1385301 0.81 SCN4A (0.51) MAPTL3MBTL1KDM4EMEN1ALDH1A1
SCHEMBL3367047 0.81 LMNA (0.53) LTA4HHAO1MAPTNPSR1KDM4E
SCHEMBL4085552 0.81 ESR2 (0.52) LTA4HMAPTKDM4EMEN1ALDH1A1
SCHEMBL6779765 0.80 SCN9A (0.54) HAO1MAPTL3MBTL1KDM4EMEN1
SCHEMBL16766999 0.79 LMNA (0.36) METAP2NOTUMMAPTMEN1KMT2A
SCHEMBL3367634 0.78 HAO1 (0.45) LTA4HHAO1MAOAMAOBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104844609-A Double-site irreversible Brutons tyrosine kinase inhibitor HANGZHOU HERTZ PHARMACEUTICAL CO LTD 2015-08-19 CN disclosed