SCHEMBL28822336

SCHEMBL28822336

N=C(N)N(C(=O)O)c1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MASP2 O00187 1/20 0.40
PLAU P00749 1/20 0.40
THPO P40225 1/20 0.40
MAPT P10636 8/20 0.39
TDP1 Q9NUW8 7/20 0.39
ALDH1A1 P00352 6/20 0.39
CYP3A4 P08684 6/20 0.39
KDM4E B2RXH2 6/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
APEX1 P27695 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
F2 P00734 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS3 P35030 1/20 0.39
ALOX15 P16050 3/20 0.37
MAPK1 P28482 2/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28826006 0.85 ALDH1A1 (0.46) MAPTTDP1ALDH1A1CYP3A4KDM4E
SCHEMBL7361311 0.83 NPSR1 (0.43) PLAUMAPTTDP1ALDH1A1CYP3A4
SCHEMBL7079951 0.82 ALDH1A1 (0.39) ALDH1A1CYP2C19RAB9ATSHRMEN1
SCHEMBL11297057 0.71 CYP3A4 (0.41) MASP2PLAUTHPOMAPTTDP1
SCHEMBL3073692 0.71 ALDH1A1 (0.45) PLAUMAPTTDP1ALDH1A1CYP3A4
SCHEMBL26108874 0.70 CYP3A4 (0.48) MAPTTDP1ALDH1A1CYP3A4KDM4E
SCHEMBL4667393 0.70 ALDH1A1 (0.44) MAPTTDP1ALDH1A1CYP3A4KDM4E
Hydrochloric Acid SCHEMBL28482173 0.69 ALDH1A1 (0.43) PLAUMAPTTDP1ALDH1A1CYP3A4
SCHEMBL10735461 0.69 LMNA (0.41) THPOMAPTALDH1A1CYP3A4KDM4E
SCHEMBL458998 0.69 ALDH1A1 (0.46) PLAUMAPTTDP1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104910047-A Preparation method of dabigatran etexilate intermediate CHANGZHOU SUNLIGHT PHARM CO LTD 2015-09-16 CN disclosed