SCHEMBL28823923

SCHEMBL28823923

Nc1ccc2c(c1)N(S(=O)(=O)c1cccs1)CCC2

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.70
ALDH1A1 P00352 3/20 0.59
NPSR1 Q6W5P4 1/20 0.59
RORC P51449 1/20 0.58
KDM4E B2RXH2 1/20 0.55
HPGD P15428 1/20 0.55
HTT P42858 1/20 0.55
RAB9A P51151 1/20 0.55
CYP11B1 P15538 1/20 0.54
CYP11B2 P19099 1/20 0.54
PKM P14618 1/20 0.46
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
BRD4 O60885 1/20 0.41
ATAD2 Q6PL18 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29817651 1.00 TSHR (0.70) TSHRALDH1A1NPSR1RORCKDM4E
SCHEMBL28823971 0.81 TSHR (0.65) TSHRALDH1A1NPSR1RORCKDM4E
SCHEMBL29817770 0.81 TSHR (0.65) TSHRALDH1A1NPSR1RORCKDM4E
SCHEMBL521211 0.76 NLRP3 (0.53) SMN1; SMN2MEN1KMT2ABRD4ATAD2
SCHEMBL29767734 0.76 NLRP3 (0.53) SMN1; SMN2MEN1KMT2ABRD4ATAD2
SCHEMBL28823950 0.74 RORC (0.57) TSHRALDH1A1NPSR1RORCKDM4E
SCHEMBL29817656 0.74 RORC (0.57) TSHRALDH1A1NPSR1RORCKDM4E
SCHEMBL28157214 0.74 RORC (0.57) TSHRALDH1A1NPSR1RORCHPGD
SCHEMBL29817735 0.74 RORC (0.57) TSHRALDH1A1NPSR1RORCHPGD
SCHEMBL4559537 0.74 KMT2A (0.59) ALDH1A1RORCCYP11B1CYP11B2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107021923-B Tetrahydroquinoline related bicyclic compound and application thereof 中国科学院广州生物医药与健康研究院 2022-09-23 CN disclosed
CN-114790169-A Tetrahydroquinoline related bicyclic compound and application thereof 中国科学院广州生物医药与健康研究院 2022-07-26 CN disclosed