SCHEMBL28823982

SCHEMBL28823982

O=C(Nc1ccc2c(c1)N(S(=O)(=O)c1ccc(F)cc1)CCO2)c1ccc(F)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.66
CPT2 P23786 3/20 0.61
CPT1A P50416 3/20 0.61
CPT1B Q92523 2/20 0.61
HTR1A P08908 1/20 0.59
HTR1D P28221 1/20 0.59
HTR1F P30939 1/20 0.59
ALDH1A1 P00352 4/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
LMNA P02545 2/20 0.57
MAPT P10636 2/20 0.57
HTT P42858 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
RAB9A P51151 1/20 0.57
CYP2C9 P11712 1/20 0.56
NR1H2 P55055 2/20 0.53
NR1H3 Q13133 2/20 0.53
NR1I2 O75469 1/20 0.53
RORA P35398 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15625873 0.86 RORC (0.68) RORCCPT2CPT1ACPT1BNR1H2
SCHEMBL5021975 0.84 RORC (0.75) RORCCPT2CPT1ACPT1BNR1H2
SCHEMBL28157203 0.82 ALDH1A1 (0.64) RORCALDH1A1MEN1KMT2ALMNA
SCHEMBL5021967 0.82 CPT1A (0.60) RORCCPT2CPT1ACPT1BMAPT
SCHEMBL5021974 0.81 CPT1A (0.56) RORCCPT2CPT1ACPT1BALDH1A1
SCHEMBL28843028 0.80 RORC (0.58) RORCCPT2CPT1ACPT1BALDH1A1
SCHEMBL5021972 0.80 CPT1A (0.58) RORCCPT2CPT1ACPT1BMAPT
SCHEMBL2001650 0.80 CNR1 (0.67) RORCCPT2CPT1ACPT1BALDH1A1
SCHEMBL755026 0.79 CPT1A (0.80) RORCCPT2CPT1ACPT1BALDH1A1
SCHEMBL1999963 0.79 CYP2C9 (0.56) RORCCPT2CPT1ACPT1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107021923-B Tetrahydroquinoline related bicyclic compound and application thereof 中国科学院广州生物医药与健康研究院 2022-09-23 CN claimed
CN-107021923-B Tetrahydroquinoline related bicyclic compound and application thereof 中国科学院广州生物医药与健康研究院 2022-09-23 CN disclosed
CN-114790169-A Tetrahydroquinoline related bicyclic compound and application thereof 中国科学院广州生物医药与健康研究院 2022-07-26 CN disclosed