Oxatomide

Oxatomide

SCHEMBL28824

O=c1[nH]c2ccccc2n1CCCN1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Oxatomide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 1/20 1.00
P2RX7 Q99572 8/20 1.00
LMNA P02545 2/20 1.00
MEN1 O00255 1/20 1.00
MLNR O43193 1/20 1.00
NR1I2 O75469 1/20 1.00
CYP1A2 P05177 1/20 1.00
CHRM2 P08172 1/20 1.00
CYP3A4 P08684 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
CYP2D6 P10635 1/20 1.00
CHRM1 P11229 1/20 1.00
CYP2C9 P11712 1/20 1.00
DRD2 P14416 1/20 1.00
PKM P14618 1/20 1.00
ADRA2C P18825 1/20 1.00
CHRM3 P20309 1/20 1.00
SLC6A2 P23975 1/20 1.00
HTR2A P28223 1/20 1.00
HTR2C P28335 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxatomide SCHEMBL29484467 1.00 P2RX7 (1.00) P2RX7LMNAMEN1MLNRNR1I2
Oxatomide SCHEMBL8693540 0.99 P2RX7 (0.98) P2RX7LMNAMEN1MLNRNR1I2
Oxatomide SCHEMBL11472510 0.99 P2RX7 (0.98) P2RX7LMNAMEN1MLNRNR1I2
Oxatomide SCHEMBL8693571 0.99 P2RX7 (0.98) P2RX7LMNAMEN1MLNRNR1I2
Oxatomide SCHEMBL7558760 0.99 P2RX7 (0.98) P2RX7LMNAMEN1MLNRNR1I2
Oxatomide SCHEMBL11199692 0.98 P2RX7 (0.95) P2RX7LMNAMEN1MLNRNR1I2
SCHEMBL11198903 0.98 P2RX7 (1.00) P2RX7LMNAMEN1MLNRNR1I2
SCHEMBL11195898 0.96 P2RX7 (1.00) P2RX7LMNAMEN1MLNRNR1I2
Water SCHEMBL11197270 0.96 P2RX7 (0.98) P2RX7LMNAMEN1MLNRNR1I2
Water SCHEMBL11197269 0.96 P2RX7 (0.98) P2RX7LMNAMEN1MLNRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4493 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
EP-4704971-A1 GAMMA STIMULATION AND NEUROMODULATOR COMBINATION THERAPY Cognito Therapeutics, Inc. (US) 2026-03-11 EP claimed
US-12569451-B2 Bio-inspired tissue-adhesive hydrogel patch and uses thereof Cellartgen Inc. (KR) 2026-03-10 US claimed
US-20250041208-A1 NEW INJECTABLE COMBINATION FORMULATION NANEXA AB (SE) 2025-02-06 US claimed
WO-2024229174-A1 GAMMA STIMULATION AND NEUROMODULATOR COMBINATION THERAPY Cognito Therapeutics, Inc. (US) 2024-11-07 WO claimed
EP-4444277-A1 NEW INJECTABLE COMBINATION FORMULATION Nanexa AB (SE) 2024-10-16 EP claimed
CN-112368300-B SPNS2 neutralizing antibodies 帝人制药株式会社 2024-10-01 CN claimed
US-20230321073-A1 COMPOSITIONS AND METHODS FOR TREATING METABOLIC DYSREGULATION Response IP Holding Company, LLC (US) 2023-10-12 US claimed
EP-4232004-A1 FRACTAL FORMULATIONS Nanogyre Sprl (BE) 2023-08-30 EP claimed
WO-2023105227-A1 NEW INJECTABLE COMBINATION FORMULATION NANEXA AB (SE) 2023-06-15 WO claimed
US-4871733-A WITH NON-STEROIDAL ANTIINFLAMMATORY ANALGESIC ASSOCIATES (US) 1989-10-03 US claimed
EP-0190449-B1 ADDITIVE-CONTAINING PAINTS OECE Industrie Chimiche Spa (IT) 1989-08-09 EP claimed
EP-0316434-A1 COUGH/COLD MIXTURES COMPRISING NON-SEDATING ANTIHISTAMINE DRUGS. SUNSHINE ABRAHAM (US) 1989-05-24 EP claimed
EP-0311677-A1 COUGH/COLD MIXTURES COMPRISING NON-SEDATING ANTIHISTAMINE DRUGS. SUNSHINE ABRAHAM (US) 1989-04-19 EP claimed
EP-0139163-B1 MULTIPLE DATA TRANSFER SYSTEM HAVING A PLURALITY OF DISK DRIVES TEAC CORPORATION (JP) 1989-04-05 EP claimed
WO-1988009656-A1 COUGH/COLD MIXTURES COMPRISING NON-SEDATING ANTIHISTAMINE DRUGS SUNSHINE ABRAHAM (US) 1988-12-15 WO claimed
WO-1988008302-A1 COUGH/COLD MIXTURES COMPRISING NON-SEDATING ANTIHISTAMINE DRUGS SUNSHINE ABRAHAM (US) 1988-11-03 WO claimed
US-4778673-A THERAPEUTIC OR PROPHYLACTIC ACTION TO PREVENT OR NEUTRALIZE IRRITATION OF RESPIRATORY TRACT MUCOSAE; TERPENES; ODORS OECE INDUSTRIE CHIMICHE SPA (IT) 1988-10-18 US claimed
EP-0190449-A1 Additive-containing paints OECE Industrie Chimiche Spa (IT) 1986-08-13 EP claimed
US-4250176-A BENZIMIDAZOLE-2-ONE, BENZOTHIAZOL-2-ONE, OR BENZOXAZOL-2-ONE SUBSTITUTIONS, ANTIANAPHALACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1981-02-10 US claimed