SCHEMBL28824003

SCHEMBL28824003

CCOC(=O)c1cnnn1-c1ccc(-c2ccccc2)c(C(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.46
ALDH1A1 P00352 11/20 0.45
SMN1; SMN2 Q16637 7/20 0.43
POLB P06746 3/20 0.43
HPGD P15428 5/20 0.43
KDM4E B2RXH2 7/20 0.43
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
HSD17B10 Q99714 3/20 0.43
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
TP53 P04637 2/20 0.43
STAT1 P42224 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MAPT P10636 4/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 3/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824000 0.88 LMNA (0.45) SCN9AALDH1A1SMN1; SMN2POLBHPGD
SCHEMBL28824024 0.85 SMN1; SMN2 (0.45) ALDH1A1SMN1; SMN2POLBHPGDKDM4E
SCHEMBL28824098 0.84 BCAT2 (0.45) SCN9AALDH1A1SMN1; SMN2HPGDKDM4E
SCHEMBL8156087 0.80 TP53 (0.58) ALDH1A1SMN1; SMN2HPGDKDM4EHSD17B10
SCHEMBL28824074 0.79 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2POLBHPGDKDM4E
SCHEMBL6765042 0.77 KDM4E (0.54) ALDH1A1SMN1; SMN2HPGDKDM4ENPC1
SCHEMBL28824021 0.77 LMNA (0.44) ALDH1A1SMN1; SMN2POLBHPGDKDM4E
SCHEMBL28823986 0.75 FOLH1 (0.44) SMN1; SMN2KDM4ENPC1RAB9AHSD17B10
SCHEMBL28824025 0.75 NPC1 (0.39) ALDH1A1SMN1; SMN2POLBHPGDNPC1
SCHEMBL8156170 0.74 IDO1 (0.46) ALDH1A1SMN1; SMN2POLBHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929676-A Heterocyclic carboxylate compounds as glycolate oxidase inhibitors 紫丁香疗法有限公司 2022-08-19 CN disclosed