SCHEMBL28824364

SCHEMBL28824364

BrCc1cccc(Oc2cccnc2)c1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.68
TDP1 Q9NUW8 1/20 0.68
TRPV6 Q9H1D0 1/20 0.52
CYP19A1 P11511 4/20 0.49
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CETP P11597 1/20 0.46
HTT P42858 1/20 0.45
GRM2 Q14416 1/20 0.45
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
MAPK1 P28482 1/20 0.43
LTA4H P09960 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4938372 0.83 LMNA (0.68) LMNATDP1TRPV6CYP19A1ALDH1A1
Pyridine SCHEMBL11782749 0.83 TRPV6 (0.52) LMNATDP1TRPV6ALDH1A1SMN1; SMN2
SCHEMBL16301357 0.83 LMNA (0.68) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL103152 0.83 LMNA (0.68) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL6201445 0.81 LMNA (0.64) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL10544332 0.80 LMNA (0.62) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL10549969 0.80 LMNA (0.62) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL22910536 0.80 LMNA (0.62) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL10223959 0.80 LMNA (0.62) LMNATDP1TRPV6CYP19A1ALDH1A1
SCHEMBL202774 0.78 ALDH1A1 (0.54) TDP1TRPV6ALDH1A1SMN1; SMN2CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805192-A Tricyclic XOR/URAT1 dual inhibitor containing 2-hydroxybenzoic acid and preparation method and application thereof 华南理工大学 2022-07-29 CN disclosed