SCHEMBL28824643

SCHEMBL28824643

COc1ccc(C=Cc2cc(C=Cc3ccc(OC)c(OC)c3)nc(O)n2)cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 4/20 0.63
PTGS1 P23219 1/20 0.63
PTGS2 P35354 1/20 0.63
APP P05067 9/20 0.60
CYP19A1 P11511 1/20 0.58
GLA P06280 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
HPGD P15428 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
CYP1B1 Q16678 3/20 0.56
TUBB4A P04350 1/20 0.56
TUBB P07437 1/20 0.56
TUBA3C P0DPH7 1/20 0.56
TUBA1B P68363 1/20 0.56
TUBA4A P68366 1/20 0.56
TUBB4B P68371 1/20 0.56
TUBB3 Q13509 1/20 0.56
TUBB2A Q13885 1/20 0.56
TUBB8 Q3ZCM7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28045186 0.82 AGTR1 (0.57) CYP1A1CYP19A1ALDH1A1MAPTHPGD
SCHEMBL9431599 0.80 CYP1A1 (0.80) CYP1A1PTGS1PTGS2APPCYP19A1
SCHEMBL9586847 0.80 CYP1A1 (0.80) CYP1A1PTGS1PTGS2APPCYP19A1
SCHEMBL28045091 0.80 PTGS2 (0.61) CYP1A1PTGS1PTGS2APPCYP19A1
SCHEMBL9173377 0.78 CYP1A1 (0.84) CYP1A1PTGS1PTGS2APPCYP19A1
SCHEMBL9173364 0.78 CYP1A1 (0.84) CYP1A1PTGS1PTGS2APPCYP19A1
SCHEMBL3396274 0.78 APP (0.74) PTGS2APPMAPTNFE2L2TTR
SCHEMBL3394666 0.78 APP (0.71) APPTUBB4ATUBBTUBA3CTUBA1B
Rhapontigenin SCHEMBL19433130 0.78 CYP1A1 (1.00) CYP1A1PTGS1PTGS2APPCYP19A1
SCHEMBL30940355 0.78 CYP1A1 (0.79) CYP1A1PTGS1PTGS2APPCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110698413-B Substituted pyrimidine derivative containing guanidyl, pharmaceutical composition thereof, and preparation method and application thereof 中国海洋大学 2023-01-24 CN claimed
CN-110698413-B Substituted pyrimidine derivative containing guanidyl, pharmaceutical composition thereof, and preparation method and application thereof 中国海洋大学 2023-01-24 CN disclosed
CN-105198820-A Substituted pyrimidine compound containing isothiourea perssad and preparation method and application thereof OCEAN UNIV CHINA 2015-12-30 CN disclosed