SCHEMBL28045091

SCHEMBL28045091

COc1ccc(C=Cc2cc(C=Cc3ccc(OC)cc3)nc(O)n2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.61
KDM4E B2RXH2 3/20 0.61
PTGS1 P23219 2/20 0.61
CYP1A1 P04798 2/20 0.61
CYP1B1 Q16678 2/20 0.61
LMNA P02545 1/20 0.61
ALOX12 P18054 1/20 0.61
MAPT P10636 1/20 0.59
NQO2 P16083 2/20 0.57
RELA Q04206 2/20 0.57
ALOX5 P09917 2/20 0.56
APP P05067 1/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
ESR1 P03372 2/20 0.55
CYP1A2 P05177 2/20 0.55
AHR P35869 2/20 0.55
ABL1 P00519 1/20 0.55
TTR P02766 1/20 0.55
ABCB1 P08183 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30219723 0.82 MEN1 (0.63) CYP1A1CYP1B1NQO2RELAAPP
SCHEMBL28824643 0.80 CYP1A1 (0.63) PTGS2PTGS1CYP1A1CYP1B1MAPT
SCHEMBL699458 0.77 RELA (0.81) PTGS2KDM4EPTGS1CYP1A1CYP1B1
SCHEMBL13790336 0.77 RELA (0.81) PTGS2KDM4EPTGS1CYP1A1CYP1B1
SCHEMBL4881152 0.77 RELA (0.81) PTGS2KDM4EPTGS1CYP1A1CYP1B1
SCHEMBL631998 0.77 RELA (0.81) PTGS2KDM4EPTGS1CYP1A1CYP1B1
SCHEMBL699457 0.77 RELA (0.81) PTGS2KDM4EPTGS1CYP1A1CYP1B1
SCHEMBL14950253 0.77 RELA (0.81) PTGS2KDM4EPTGS1CYP1A1CYP1B1
SCHEMBL3394328 0.76 APP (0.62) PTGS2KDM4EPTGS1CYP1A1CYP1B1
Resveratrol 4'-Methyl Ether SCHEMBL563262 0.76 PTGS2 (1.00) PTGS2KDM4EPTGS1CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110698413-B Substituted pyrimidine derivative containing guanidyl, pharmaceutical composition thereof, and preparation method and application thereof 中国海洋大学 2023-01-24 CN claimed
CN-110698413-B Substituted pyrimidine derivative containing guanidyl, pharmaceutical composition thereof, and preparation method and application thereof 中国海洋大学 2023-01-24 CN disclosed
CN-105198820-B A kind of substituted pyrimidines compound of the group containing isothiourea and its preparation method and application 中国海洋大学 2019-10-01 CN disclosed
CN-105198820-A Substituted pyrimidine compound containing isothiourea perssad and preparation method and application thereof OCEAN UNIV CHINA 2015-12-30 CN disclosed