SCHEMBL28824792

SCHEMBL28824792

CC(C)COC(=O)NC(Cc1ccc2ccccc2n1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
NR3C2 P08235 1/20 0.41
CYSLTR2 Q9NS75 5/20 0.41
CYSLTR1 Q9Y271 5/20 0.41
ELANE P08246 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
MAOB P27338 1/20 0.40
CASP3 P42574 3/20 0.39
CASP7 P55210 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PRNP P04156 1/20 0.39
MAPK10 P53779 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29858123 1.00 CYP1A2 (0.45) CYP1A2NR3C2CYSLTR2CYSLTR1ELANE
SCHEMBL29858159 0.88 KMT2A (0.49) CYP1A2CYSLTR2CYSLTR1SIRT2KDM4E
SCHEMBL21467795 0.88 KMT2A (0.49) CYP1A2CYSLTR2CYSLTR1SIRT2KDM4E
SCHEMBL28824795 0.88 KMT2A (0.49) CYP1A2CYSLTR2CYSLTR1SIRT2KDM4E
SCHEMBL28824775 0.87 CYP1A2 (0.47) CYP1A2CYSLTR2CYSLTR1SIRT2
SCHEMBL21467676 0.87 CYP1A2 (0.47) CYP1A2CYSLTR2CYSLTR1SIRT2
SCHEMBL29858135 0.87 CYP1A2 (0.47) CYP1A2CYSLTR2CYSLTR1SIRT2
SCHEMBL28824786 0.85 CASP3 (0.47) CYP1A2CYSLTR2CYSLTR1CASP3CASP7
SCHEMBL29858069 0.85 CASP3 (0.47) CYP1A2CYSLTR2CYSLTR1CASP3CASP7
SCHEMBL19407482 0.83 GABRB1 (0.45) CYP1A2CYSLTR2CYSLTR1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563045-B Pd (II) -catalysed enantioselective beta-methylene C (sp) 3 ) -H bond activation 斯克里普斯研究学院 2022-08-23 CN disclosed