SCHEMBL28825571

SCHEMBL28825571

Cc1ncc(Cn2ccc(-c3ccc(F)c(F)c3)n2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
CACNA1G O43497 4/20 0.42
CACNA1H O95180 4/20 0.42
CACNA1I Q9P0X4 4/20 0.42
KDM1A O60341 3/20 0.41
HDAC1 Q13547 3/20 0.41
GRM2 Q14416 1/20 0.40
ALDH1A1 P00352 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 4/20 0.39
KDM4E B2RXH2 4/20 0.39
LMNA P02545 3/20 0.39
HPGD P15428 3/20 0.39
RAB9A P51151 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825461 0.84 CYP11B1 (0.51) CYP11B1CYP11B2MAPTSMN1; SMN2CACNA1G
SCHEMBL28949586 0.83 KDM4E (0.45) CYP11B1MAPTSMN1; SMN2CACNA1GCACNA1H
SCHEMBL28825651 0.82 GRIN1 (0.52) CYP11B1CYP11B2MAPTSMN1; SMN2CACNA1G
SCHEMBL28825447 0.79 GRIN2B (0.50) CYP11B1CYP11B2MAPTSMN1; SMN2ALDH1A1
SCHEMBL28825580 0.79 GRIN1 (0.43) CYP11B1CYP11B2MAPTSMN1; SMN2KDM1A
SCHEMBL28949561 0.77 GRIN2B (0.54) CYP11B1CYP11B2MAPTSMN1; SMN2KDM1A
SCHEMBL28825563 0.76 GRIN1 (0.53) CYP11B1CYP11B2MAPTSMN1; SMN2CACNA1G
SCHEMBL28825546 0.76 GRIN2B (0.53) CYP11B1CYP11B2MAPTSMN1; SMN2CACNA1G
SCHEMBL28825694 0.75 GRIN1 (0.42) CYP11B1CYP11B2MAPTSMN1; SMN2CACNA1G
SCHEMBL28825484 0.73 GRIN1 (0.43) MAPTSMN1; SMN2KDM1AHDAC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed