SCHEMBL28825573

SCHEMBL28825573

Cc1ncc(Cn2cccn2)c(-c2ccc(F)c(F)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 7/20 0.41
GRIN1 Q05586 6/20 0.39
PDE4B Q07343 2/20 0.38
KLKB1 P03952 2/20 0.37
KLK7 P49862 1/20 0.36
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
BRD4 O60885 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
USP2 O75604 3/20 0.34
CYP1A2 P05177 3/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2C9 P11712 2/20 0.34
MAPK1 P28482 2/20 0.34
CYP2C19 P33261 2/20 0.34
TSHR P16473 1/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949587 0.83 GRIN2B (0.40) GRIN2BGRIN1PDE4BKLKB1GAA
SCHEMBL28825565 0.80 GRIN2B (0.43) GRIN2BGRIN1KLKB1KLK7GAA
SCHEMBL28825448 0.78 GAA (0.47) GRIN2BGRIN1PDE4BKLKB1KLK7
SCHEMBL28825653 0.78 GAA (0.44) GRIN2BGRIN1PDE4BKLKB1GAA
SCHEMBL28825549 0.76 GRIN2B (0.40) GRIN2BGRIN1PDE4BKLKB1KLK7
SCHEMBL28949563 0.75 PDE4B (0.46) GRIN2BGRIN1PDE4BGAAMAPT
SCHEMBL28825445 0.73 GRIN2B (0.51) GRIN2BGRIN1KLKB1CYP1A2CYP2C9
SCHEMBL28825510 0.71 GRIN2B (0.52) GRIN2BGRIN1KLKB1GAAMAPT
SCHEMBL28825487 0.71 GRIN2B (0.51) GRIN2BGRIN1KLKB1GAAMAPT
SCHEMBL1457252 0.68 GAA (0.51) KLKB1GAAMAPTTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed