SCHEMBL28825549

SCHEMBL28825549

Cc1nc(-c2ccc(F)c(F)c2)ccc1Cn1cccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.40
GRIN1 Q05586 3/20 0.40
KLKB1 P03952 3/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
BRD4 O60885 1/20 0.36
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
NSD2 O96028 1/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
KMO O15229 1/20 0.35
KLK7 P49862 1/20 0.35
TRPV3 Q8NET8 2/20 0.35
PDE4B Q07343 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825615 0.92 GRIN2B (0.46) GRIN2BGRIN1KLKB1BRD4PRKACA
SCHEMBL28825565 0.80 GRIN2B (0.43) GRIN2BGRIN1KLKB1CYP11B1CYP11B2
SCHEMBL28825573 0.76 GRIN2B (0.41) GRIN2BGRIN1KLKB1CYP11B1CYP11B2
SCHEMBL28825642 0.74 GRIN2B (0.46) GRIN2BGRIN1PDE4B
SCHEMBL28825445 0.72 GRIN2B (0.51) GRIN2BGRIN1KLKB1
SCHEMBL28825476 0.72 GRIN2B (0.49) GRIN2BGRIN1ALDH1A1LMNAPDE4B
SCHEMBL31172834 0.72 GAA (0.51) KLKB1BRD4PDE4BCA12CA1
SCHEMBL28825546 0.71 GRIN2B (0.53) GRIN2BGRIN1CYP11B1CYP11B2ALDH1A1
SCHEMBL28825448 0.70 GAA (0.47) GRIN2BGRIN1KLKB1CYP11B1CYP11B2
SCHEMBL28825653 0.70 GAA (0.44) GRIN2BGRIN1KLKB1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed