SCHEMBL28825445

SCHEMBL28825445

Cc1cc(-c2cc(C)c(Cn3cccn3)cn2)ccc1F

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 14/20 0.51
GRIN1 Q05586 8/20 0.42
KCNH2 Q12809 6/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
KLKB1 P03952 1/20 0.38
SRC P12931 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825565 0.93 GRIN2B (0.43) GRIN2BGRIN1KLKB1
SCHEMBL28949569 0.84 GRIN2B (0.38) GRIN2BGRIN1KCNH2KLKB1
SCHEMBL28825483 0.81 GRIN2B (0.44) GRIN2BGRIN1
SCHEMBL28825615 0.81 GRIN2B (0.46) GRIN2BGRIN1KCNH2CYP1A2CYP2C9
SCHEMBL28825510 0.77 GRIN2B (0.52) GRIN2BGRIN1KCNH2CYP1A2CYP2C9
SCHEMBL28825487 0.76 GRIN2B (0.51) GRIN2BGRIN1KCNH2CYP1A2CYP2C9
SCHEMBL28825573 0.73 GRIN2B (0.41) GRIN2BGRIN1CYP1A2CYP2C9CYP2C19
SCHEMBL28825549 0.72 GRIN2B (0.40) GRIN2BGRIN1KLKB1
SCHEMBL28028438 0.68 MAPT (0.35) GRIN2BGRIN1CYP1A2KLKB1
SCHEMBL14822759 0.68 RIPK1 (0.44) GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed