SCHEMBL28825583

SCHEMBL28825583

Cc1cncc([CH]c2ccc(Cl)c(OC(F)F)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 16/20 0.44
GRIN1 Q05586 13/20 0.44
RXRA P19793 11/20 0.38
KCNH2 Q12809 8/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949605 0.86 GRIN2B (0.42) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825625 0.85 GRIN1 (0.43) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825657 0.85 GRIN2B (0.43) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825617 0.85 GRIN2B (0.46) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825527 0.83 GRIN2B (0.44) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825534 0.83 GRIN2B (0.44) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825640 0.76 GRIN2B (0.47) GRIN2BGRIN1RXRAKCNH2
SCHEMBL900483 0.71 MEN1 (0.52) GRIN2BGRIN1RXRAKCNH2
SCHEMBL28825624 0.71 GRIN2B (0.39) GRIN2BGRIN1RXRAKCNH2
SCHEMBL10914962 0.70 ALDH1A1 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed