SCHEMBL288260

SCHEMBL288260

O=C(O)[C@H]1Cc2ccccc2CN1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
EGLN1 Q9GZT9 1/20 0.52
PRCP P42785 1/20 0.52
OPRM1 P35372 1/20 0.48
OPRD1 P41143 1/20 0.48
OPRK1 P41145 1/20 0.48
PNMT P11086 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29350565 1.00 GAA (0.58) GAAMAPTMEN1KMT2AEGLN1
SCHEMBL29398238 1.00 GAA (0.58) GAAMAPTMEN1KMT2AEGLN1
SCHEMBL29350888 1.00 GAA (0.58) GAAMAPTMEN1KMT2AEGLN1
SCHEMBL288272 1.00 GAA (0.58) GAAMAPTMEN1KMT2AEGLN1
SCHEMBL43168 1.00 GAA (0.58) GAAMAPTMEN1KMT2AEGLN1
Bromide SCHEMBL8763315 0.98 GAA (0.56) GAAMAPTMEN1KMT2AEGLN1
Hydrochloric Acid SCHEMBL7272493 0.98 GAA (0.56) GAAMAPTMEN1KMT2AEGLN1
Hydrochloric Acid SCHEMBL1202518 0.98 GAA (0.56) GAAMAPTMEN1KMT2AEGLN1
Hydrochloric Acid SCHEMBL32677098 0.98 GAA (0.56) GAAMAPTMEN1KMT2AEGLN1
SCHEMBL28412655 0.98 GAA (0.56) GAAMAPTMEN1KMT2AEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 259 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111254180-B Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by enzymatic resolution 浙江大学 2023-04-28 CN claimed
CN-111254170-B Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by multienzyme coupling 浙江大学 2023-04-28 CN claimed
CN-111254170-A Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by multi-enzyme coupling 浙江大学 2020-06-09 CN claimed
CN-105007928-A Synthetic linear apelin mimetics for the treatment of heart failure NOVARTIS AG 2015-10-28 CN claimed
EP-2462147-B1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2014-11-12 EP claimed
EP-0902781-B1 PREPARATION OF (S)-DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID T-BUTYLAMIDE PCBU SERVICES INC (US) 2003-12-17 EP claimed
US-20020072604-A1 Melanocortin receptor ligands CARPINO PHILIP A (US) 2002-06-13 US claimed
EP-0902781-A4 PREPARATION OF (S)-DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID T-BUTYLAMIDE NSC TECHNOLOGIES LLC (US) 2000-07-19 EP claimed
EP-0902781-A1 PREPARATION OF (S)-DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID T-BUTYLAMIDE Monsanto Company (US) 1999-03-24 EP claimed
WO-1997030976-A1 PREPARATION OF (S)-DECAHYDROISOQUINOLINE-3-CARBOXYLIC ACID T-BUTYLAMIDE MONSANTO COMPANY (US) 1997-08-28 WO claimed
US-5587481-A Preparation of (S)-decahydroisoquinoline-3-carboxylic acid t-butylamide THE MONSANTO COMPANY (US) 1996-12-24 US claimed
US-20260083852-A1 PROTEOGLYCAN MIMETICS FOR ENHANCED WOUND HEALING, ANGIOGENESIS, AND VASCULAR REPAIR UNIV CALIFORNIA (US) 2026-03-26 US disclosed
US-12485182-B2 Proteoglycan mimetics for enhanced wound healing, angiogenesis, and vascular repair THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-12-02 US disclosed
US-20250353875-A1 PEPTIDE SYNTHESIS METHOD FOR SUPPRESSING DEFECT CAUSED BY DIKETOPIPERAZINE FORMATION CHUGAI PHARMACEUTICAL CO LTD (JP) 2025-11-20 US disclosed
EP-4509517-A1 PEPTIDE SYNTHESIS METHOD FOR SUPPRESSING DEFECT CAUSED BY DIKETOPIPERAZINE FORMATION CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2025-02-19 EP disclosed
EP-0845464-A2 S type 2-substituted hydroxy-2-indolidinylbutyric ester compounds as intermediates for camptothecin derivatives TANABE SEIYAKU CO., LTD. (JP) 1998-06-03 EP disclosed
CN-1165817-A Novel metalloprotease inhibitors, process for preparing them and pharmaceutical compositions containing them ADIR (FR) 1997-11-26 CN disclosed
WO-1997017050-A3 AN IMPROVED METHOD FOR PREPARATION OF SUBSTITUTED TETRAHYDROISOQUINOLINES MONSANTO CO (US) 1997-06-05 WO disclosed
WO-1997017050-A2 AN IMPROVED METHOD FOR PREPARATION OF SUBSTITUTED TETRAHYDROISOQUINOLINES MONSANTO COMPANY (US) 1997-05-15 WO disclosed
WO-1997017050-A2 AN IMPROVED METHOD FOR PREPARATION OF SUBSTITUTED TETRAHYDROISOQUINOLINES MONSANTO COMPANY (US) 1997-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020072604-A1 Melanocortin receptor ligands MC1R, MC4R, MC3R GAA 3810/4885MAPT 3509/4885MEN1 770/4885
US-12485182-B2 Proteoglycan mimetics for enhanced wound healing, angiogenesis, and vascular repair PDGFA, PDGFRB, TEK GAA 818/4885MAPT 3707/4885MEN1 4811/4885
US-20260083852-A1 PROTEOGLYCAN MIMETICS FOR ENHANCED WOUND HEALING, ANGIOGENESIS, AND VASCULAR REPAIR PDGFA, DCLRE1A, PDGFRA GAA 2925/4885MAPT 4854/4885MEN1 4697/4885
US-20250353875-A1 PEPTIDE SYNTHESIS METHOD FOR SUPPRESSING DEFECT CAUSED BY DIKETOPIPERAZINE FORMATION VIP, NPPA, DNPEP GAA 1505/4885MAPT 4114/4885MEN1 162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.