SCHEMBL28826604

SCHEMBL28826604

O=C1c2ccccc2Cc2cccc(Cc3ccncc3)c21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.47
CYP19A1 P11511 8/20 0.47
TNF P01375 3/20 0.47
CHRM2 P08172 2/20 0.43
CHRM4 P08173 2/20 0.43
CHRM5 P08912 2/20 0.43
CHRM1 P11229 2/20 0.43
CHRM3 P20309 1/20 0.43
BCHE P06276 1/20 0.41
CES1 P23141 1/20 0.41
KCNQ2 O43526 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
CYP11B2 P19099 2/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9719382 0.99 TNF (0.48) MAOACYP19A1TNFCHRM2CHRM4
SCHEMBL27640476 0.90 MAOA (0.52) MAOABCHECES1CYP1A2CYP3A4
SCHEMBL10517737 0.85 CYP19A1 (0.44) MAOACYP19A1TNFCHRM2CHRM4
SCHEMBL27640284 0.84 MAOA (0.46) MAOABCHECES1CYP1A2MIF
SCHEMBL27431850 0.83 KCNQ2 (0.46) MAOACYP19A1TNFBCHECES1
SCHEMBL27640287 0.80 MAOA (0.44) MAOABCHECES1MIFMAPK1
SCHEMBL10447390 0.79 MAOA (0.57) MAOACYP19A1TNFBCHECES1
SCHEMBL28562503 0.78 PNMT (0.57) CYP19A1TNFCHRM2CHRM4CHRM5
SCHEMBL27661033 0.78 CALM1 (0.45) MAOAPKM
SCHEMBL17715427 0.77 MAOA (0.55) MAOACYP19A1TNFBCHECES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115702141-A Cyclobutyl-urea derivatives 爱杜西亚药品有限公司 2023-02-14 CN disclosed
CN-115461327-A Spiro urea derivatives 爱杜西亚药品有限公司 2022-12-09 CN disclosed
CN-108884030-B Improved labeling of nucleophiles using bipyridines 安捷伦科技有限公司 2022-06-28 CN disclosed