SCHEMBL28828024

SCHEMBL28828024

NC(=O)c1cc2cccc(-c3ccc(OC(F)(F)F)cc3)c2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.42
TPX2 Q9ULW0 1/20 0.42
CHEK1 O14757 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
SCN9A Q15858 9/20 0.42
ABL1 P00519 2/20 0.41
CHEK2 O96017 1/20 0.41
P2RY1 P47900 1/20 0.40
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
KIT P10721 1/20 0.39
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064557 0.84 HDAC11 (0.47) SCN9ACHEK2
SCHEMBL24074547 0.82 GRM2 (0.44) KMT2ACHEK2FLT3
SCHEMBL16571054 0.81 NTRK1 (0.40) AURKATPX2CHEK1KDM4EGAA
SCHEMBL16571279 0.80 KDM4E (0.39) AURKATPX2CHEK1KDM4EGAA
SCHEMBL30494484 0.80 HPGD (0.46) KDM4EKMT2A
SCHEMBL28064535 0.80 HPGD (0.46) KDM4EKMT2A
SCHEMBL28064654 0.78 IKBKB (0.39) KMT2A
SCHEMBL28207999 0.76 KDM4E (0.60) AURKATPX2KDM4EGAAKMT2A
SCHEMBL28064616 0.73 HRH4 (0.40) KMT2A
SCHEMBL4860862 0.72 KDM4E (0.73) KDM4EGAAKMT2AFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555763-A Indole-carboxamide derivatives HOFFMANN LA ROCHE 2016-05-04 CN claimed
CN-105555763-A Indole-carboxamide derivatives HOFFMANN LA ROCHE 2016-05-04 CN disclosed