SCHEMBL28828408

SCHEMBL28828408

COCCOc1ccc(-c2ccc3c(c2)C(OC(N)=O)C(C)(C)C3)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.41
CHEK1 O14757 3/20 0.39
S1PR1 P21453 1/20 0.38
PPARG P37231 2/20 0.37
RARG P13631 3/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
BTK Q06187 1/20 0.34
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
BACE1 P56817 6/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828573 0.92 CHEK1 (0.41) CHEK2CHEK1S1PR1PPARGRARG
SCHEMBL29228189 0.90 S1PR1 (0.41) CHEK2CHEK1S1PR1PPARGRARG
SCHEMBL28828521 0.83 CHEK1 (0.46) CHEK2CHEK1
SCHEMBL29228373 0.83 S1PR1 (0.41) CHEK2CHEK1S1PR1PPARGRARG
SCHEMBL28828381 0.82 KIF11 (0.34) RARGRARARARB
SCHEMBL28828488 0.82 ACACB (0.37) RARARARB
SCHEMBL28828372 0.82 RARB (0.40) RARARARB
SCHEMBL28828438 0.82 FYN (0.40) CHEK2CHEK1RARGRARARARB
SCHEMBL28828548 0.81 KDM4E (0.38) BACE1OPRM1
SCHEMBL28950173 0.81 KLKB1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed