SCHEMBL28828573

SCHEMBL28828573

COCCOc1ccc(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.41
CHEK2 O96017 2/20 0.41
S1PR1 P21453 1/20 0.38
CRBN Q96SW2 1/20 0.35
PPARG P37231 2/20 0.35
PPARD Q03181 4/20 0.34
RARA P10276 2/20 0.34
RARB P10826 2/20 0.34
RARG P13631 1/20 0.34
BTK Q06187 1/20 0.34
FFAR1 O14842 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
KIT P10721 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828521 0.92 CHEK1 (0.46) CHEK1CHEK2FFAR1FFAR4NR4A2
SCHEMBL28828408 0.92 CHEK2 (0.41) CHEK1CHEK2S1PR1PPARGRARA
SCHEMBL28828438 0.90 FYN (0.40) CHEK1CHEK2PPARDRARARARB
SCHEMBL28828488 0.90 ACACB (0.37) PPARDRARARARB
SCHEMBL28828372 0.90 RARB (0.40) PPARDRARARARB
SCHEMBL29228373 0.90 S1PR1 (0.41) CHEK1CHEK2S1PR1CRBNPPARG
SCHEMBL28828468 0.89 PARP1 (0.36) CRBNPPARGPPARDRARARARB
SCHEMBL28828590 0.88 PARP10 (0.39) CHEK2PPARD
SCHEMBL29121247 0.88 PARP10 (0.39) CHEK2PPARD
SCHEMBL28828363 0.87 CHRNB2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed