SCHEMBL28828663

SCHEMBL28828663

COc1cc2c(cc1-c1cccc(OC(C)C)c1)CC(C)(C)C2OC(N)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
FFAR4 Q5NUL3 2/20 0.34
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
DHODH Q02127 1/20 0.34
SLC16A3 O15427 1/20 0.33
SLC16A1 P53985 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2E1 P05181 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828506 0.92 CYP1A1 (0.40) DHODHHSP90AA1HSP90AB1CYP1A1CYP1A2
SCHEMBL28828687 0.90 ERN1 (0.36) FFAR4BACE1
SCHEMBL28828597 0.89 PRMT5 (0.37) DHODHSLC16A3SLC16A1
SCHEMBL28828451 0.88 CTSA (0.38) RXRARXRBAKR1C3AKR1C2
SCHEMBL28828689 0.88 RXRA (0.37) RXRARXRBDHODHMAPT
SCHEMBL28828494 0.87 KDM1A (0.39) RXRARXRBFFAR4AKR1C3AKR1C2
SCHEMBL29121218 0.87 KDM1A (0.39) RXRARXRBFFAR4AKR1C3AKR1C2
SCHEMBL28828636 0.86 ERN1 (0.41) DHODHALDH1A1LMNAMAPTHPGD
SCHEMBL28828464 0.85 F2R (0.39) CYP1A2LMNA
SCHEMBL28828656 0.85 RXRA (0.46) RXRARXRBFFAR4DHODHHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed